Novel phenylamino acetamide derivatives as potent and selective κ opioid receptor agonistsCHU, Guo-Hua; MINGHUA GU; DOLLE, Roland E et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 3, pp 645-648, issn 0960-894X, 4 p.Article

Indolyl and dihydroindolyl N-glycinamides as potent and in vivo active NPY5 antagonistsLINGYUN WU; KAI LU; PACKIARAJAN, Mathivanan et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 6, pp 2167-2171, issn 0960-894X, 5 p.Article

Direct Fmoc-Chemistry-Based Solid-Phase Synthesis of Peptidyl ThioestersSHARMA, Indrajeet; CRICH, David.Journal of organic chemistry. 2011, Vol 76, Num 16, pp 6518-6524, issn 0022-3263, 7 p.Article

Bifunctional agents for reperfusion arrhythmias: Novel hybrid vitamin E/class I antiarrhythmicsKOUFAKI, Maria; CALOGEROPOULOU, Theodora; REKKA, Eleni et al.Bioorganic & medicinal chemistry. 2003, Vol 11, Num 23, pp 5209-5219, issn 0968-0896, 11 p.Article

Physicochemical determinants of passive membrane permeability : Role of solute hydrogen-bonding potential and volumeGOODWIN, Jay T; CONRADI, Robert A; HO, Norman F. H et al.Journal of medicinal chemistry (Print). 2001, Vol 44, Num 22, pp 3721-3729, issn 0022-2623Article

A bivalent ligand (KMN-21) antagonist for μ/κ heterodimeric opioid receptorsSHIJUN ZHANG; YEKKIRALA, Ajay; YE TANG et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 24, pp 6978-6980, issn 0960-894X, 3 p.Article

Discovery of Disubstituted Cyclohexanes as a New Class of CC Chemokine Receptor 2 AntagonistsCHERNEY, Robert J; RUOWEI MO; SOLOMON, Kimberly A et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 4, pp 721-724, issn 0022-2623, 4 p.Article

An efficient and versatile synthesis of acylpolyamine spider toxinsNIHEI, Ken-Ichi; KATO, Massuo J; YAMANE, Tetsuo et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 3, pp 299-302, issn 0960-894XArticle

Novel sulfone-containing di- and trisubstituted cyclohexanes as potent CC chemokine receptor 2 (CCR2) antagonistsCHERNEY, Robert J; RUOWEI MO; DECICCO, Carl P et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 13, pp 3418-3422, issn 0960-894X, 5 p.Article

Identification of Lead Compounds As Antagonists of Protein Bcl-x_L with a Diversity-Oriented Multidisciplinary ApproachDI MICCO, Simone; VITALE, Romina; PELLECCHIA, Maurizio et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 23, pp 7856-7867, issn 0022-2623, 12 p.Article

Characterization of the binding properties of SIRT2 inhibitors with a N-(3-phenylpropenoyl)-glycine tryptamide backboneKIVIRANTA, Päivi H; SALO, Heikki S; WALLEN, Erik A. A et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 17, pp 8054-8062, issn 0968-0896, 9 p.Article

Discovery of INCB3344, a potent, selective and orally bioavailable antagonist of human and murine CCR2XUE, Chu-Biao; ANLAI WANG; ANAND, Rajan et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 24, pp 7473-7478, issn 0960-894X, 6 p.Article

Design, synthesis and cell growth inhibitory activity of a series of novel aminosubstituted xantheno[1,2-d]imidazoles in breast cancer cellsKOSTAKIS, Ioannis K; POULI, Nicole; MARAKOS, Panagiotis et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 6, pp 3445-3455, issn 0968-0896, 11 p.Article

Synthesis and anticonvulsant activity of a class of 2-amino 3-hydroxypropanamide and 2-aminoacetamide derivativesGHIDINI, Eleonora; DELCANALE, Maurizio; BERGAMASCHI, Marco et al.Bioorganic & medicinal chemistry. 2006, Vol 14, Num 10, pp 3263-3274, issn 0968-0896, 12 p.Article

Structure-based discovery of nonpeptidic small organic compounds to block the T cell response to myelin basic proteinKOEHLER, Niklas K. U; YANG, Chao-Yie; LONG, Ya-Qiu et al.Journal of medicinal chemistry (Print). 2004, Vol 47, Num 21, pp 4989-4997, issn 0022-2623, 9 p.Article

5,7,8-Trimethyl-benzopyran and 5,7,8-Trimethyl-1,4-benzoxazine Aminoamide Derivatives as Novel Antiarrhythmics against Ischemia-Reperfusion InjuryKOINI, Eftychia N; PAPAZAFIRI, Panagiota; VASSILOPOULOS, Athanasios et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 8, pp 2328-2340, issn 0022-2623, 13 p.Article

Cyclopentane-based human NK1 antagonists. Part 2: Development of potent, orally active, water-soluble derivativesMEURER, Laura C; FINKE, Paul E; CHICCHI, Gary G et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 17, pp 4504-4511, issn 0960-894X, 8 p.Article

A molecular basis for the selectivity of thiadiazole urea inhibitors with stromelysin-1 and gelatinase-a from Generalized Born molecular dynamics simulationsRIZZO, Robert C; TOBA, Samuel; KUNTZ, Irwin D et al.Journal of medicinal chemistry (Print). 2004, Vol 47, Num 12, pp 3065-3074, issn 0022-2623, 10 p.Article

Cationic lipids containing protonated cyclen and different hydrophobic groups linked by uracil-PNA monomer: Synthesis and application for gene deliveryLIU, Jun-Liang; MA, Qing-Ping; HUANG, Qing-Dong et al.European journal of medicinal chemistry. 2011, Vol 46, Num 9, pp 4133-4141, issn 0223-5234, 9 p.Article

Acylglycinamides as inhibitors of glycine transporter type 1BLUNT, Richard; PORTER, Roderick; GORDON, Laurie et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 20, pp 6176-6179, issn 0960-894X, 4 p.Article

Synthesis and structure-activity relationship of imidazo (1,2 -a )thieno (3,2 -e )pyrazines as IKK-β inhibitorsBELEMA, Makonen; BUNKER, Amy; PATTOLI, Mark A et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 15, pp 4284-4289, issn 0960-894X, 6 p.Article

Synthesis and biological evaluation of technetium-99m-labeled deoxyglucose derivatives as imaging agents for tumorXIANGJI CHEN; LIANG LI; FEI LIU et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 21, pp 5503-5506, issn 0960-894X, 4 p.Article

Preparation of a technetium-99m SPECT agent for imaging the sigma-2 receptor status of solid tumorsMACH, Robert H; WHEELER, Kenneth T; BLAIR, Suwanna et al.Journal of labelled compounds & radiopharmaceuticals. 2001, Vol 44, Num 13, pp 899-908, issn 0362-4803Conference Paper

Non-depolarizing neuromuscular blocking activity of bisquaternary amino di- and tripeptide derivativesBOOIJ, Leo H. D. J; VAN DER BROEK, Leon A. G. M; CAULFIELD, Wilson et al.Journal of medicinal chemistry (Print). 2000, Vol 43, Num 25, pp 4822-4833, issn 0022-2623Article

Design and synthesis of a siderophore conjugate as a potent PSMA inhibitor and potential diagnostic agent for prostate cancerPINGYU DING; HELQUIST, Paul; MILLER, Marvin J et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 4, pp 1648-1657, issn 0968-0896, 10 p.Article